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Top publikace

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Cankařová, N.; Krchňák, V.
Regioselective Cyclic Iminium Formation of Ugi Advanced Intermediates: Rapid Access to 3,4-Dihydropyrazin-2(1H)-ones and Other Diverse Nitrogen-Containing Heterocycles
Molecules 2023, 28 (7), 3062 (1-17). DOI: 10.3390/molecules28073062



Tomanová, M.; Vaňková, I.; Toman, D.; Přibylka, A.; Nemec, I.; Cankař, P.
Axially Chiral Sulfonic Acids for Brønsted Acid Catalysis: 8-Benzoimidazolylnaphthalene-1-sulfonic Acids and Their Derivatives
J. Org. Chem. 2023, 88 (13), 9265–9276. DOI: 10.1021/acs.joc.3c00818


Ondrová, K.; Zůvalová, I.; Vyhlídalová, B.; Krasulová, K.; Miková, E.; Vrzal, R.; Nádvorník, P.; Nepal, B.; Kortagere, S.; Kopečná, M.; Kopečný, D.; Šebela, M.; Rastinejad, F.; Pu, H.; Soural, M.; Rolfes, K. M.; Haarmann-Stemmann, T.; Li, H.; Mani, S.; Dvořák, Z.
Monoterpenoid aryl hydrocarbon receptor allosteric antagonists protect against ultraviolet skin damage in female mice
Nat. Commun. 2023, 14 (-), 2728-2743. DOI: 10.1038/s41467-023-38478-6


Krajcovicova, S.; Spring, D. R.
Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late-Stage Functionalisation
Angew. Chem. Int. Ed. 2023, e202307782 (-), -. DOI: 10.1002/anie.202307782


King, T.; Walsh, S.; Kapun, M.; Wharton, T.; Krajcovicova, S.; Glossop, M.; Spring, D.
Disulfide re-bridging reagents for single-payload antibody-drug conjugates
Chemical Communications 2023, (-), -. DOI: 10.1039/D3CC02980H


Šamšulová, V.; Šedivá, M.; Kóňa, J. ; Klaudiny, J.; Poláková, M.
A Comparison of the Antibacterial Efficacy of Carbohydrate Lipid‐like (Thio)Ether, Sulfone, and Ester Derivatives against Paenibacillus larvae
Molecules 2023, 28 (-), 2516. DOI: doi.org/10.3390/molecules28062516