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Schütznerová, E.; Oliver, A.; Slough, G. A.; Krchňák, V.
Traceless Solid-Phase Synthesis of Fused Chiral Macrocycles via Conformational Constraint-Assisted Cyclic Iminium Formation
Chem. Eur. J. 2017, 21 (37), 12876-12885. DOI: 10.1002/chem.201702461

Přibylka, A.; Krchňák, V.
Gold-Catalyzed Solid-Phase Synthesis of 3,4-Dihydropyrazin-2(1H)-ones: Relevant Pharmacophores and Peptide Backbone Constraints
ACS Comb. Sci. 2017, 19 (11), 681-686. DOI: 10.1021/acscombsci.7b00117

Schütznerová, E.; Krchňák, V.
Intramolecular Arylation of 2-Nitrobenzenesulfonamides: A Route to Diverse Nitrogenous Heterocycles
Top. Heterocycl. Chem. 2017, 52 (-), 139-166. DOI: 10.1007/7081_2016_5

Kloss, F.; Krchňák, V.; Krchňáková, A.; Schieferdecker, S.; Dreisbach, J.; Krone, V.; Möllmann, U.; Hoelscher, M.; Miller, M. J.
In Vivo Dearomatization of the Potent Antituberculosis Agent BTZ043 via Meisenheimer Complex Formation
Angew. Chem. Int. Ed. 2017, 56 (8), 2187-2191. DOI: 10.1002/anie.201609737

Krchňák, V. (editor)
Solid-Phase Synthesis of Nitrogenous Heterocycles in Topics in Heterocyclic Chemistry
kniha, Springer, 2017. DOI:

Schütznerová, E.; Oliver, A. G.; Slough, G. A.; Krchňák, V.
Traceless Solid-Phase Synthesis of Fused Chiral Macrocycles via Conformational Constraint-Assisted Cyclic Iminium Formation
„2nd International Caparica Christmas Congress on Translational Chemistry“ (IC3TC 2017), December 4-7, 2017, Largo Aldeia dos Capuchos, Caparica (Portugalsko), poster . DOI:

Přibylka, A.; Krchňák, V.
Gold-Catalyzed Polymer-Supported Synthesis of Diversely Substituted 3,4-Dihydropyrazin-2(1H)-ones for Applications in Drug Discovery and Peptide Backbone Constraints
„2nd International Caparica Christmas Congress on Translational Chemistry“ (IC3TC 2017), December 4-7, 2017, Largo Aldeia dos Capuchos, Caparica (Portugalsko), poster . DOI:

Carbain, B.; Schütznerová, E.; Přibylka, A.; Krchňák, V.
Solid-Phase Synthesis of 3,4-Dihydroquinoxalin-2(1H)-ones via the Cyclative Cleavage of N-Arylated Carboxamides
Adv. Synth. Catal. 2016, 358 (5), 701-706. DOI: 10.1002/adsc.201500826

Schütznerová, E.; Krchňák, V.
N-Oxide as an Intramolecular Oxidant in the Baeyer-Villiger Oxidation: Synthesis of 2-Alkyl-2H-indazol-3-yl Benzoates and 2-Alkyl-1,2-dihydro-3H-indazol-3-ones
J. Org. Chem. 2016, 81 (9), 3585-3596. DOI: 10.1021/acs.joc.6b00251

La-Venia, A.; Medran, N. S.; Krchňák, V.; Testero, S. A.
Synthesis of a Small Library of Imidazolidin-2-ones using Gold Catalysis on Solid Phase
ACS Comb. Sci. 2016, 18 (8), 482-489. DOI: 10.1021/acscombsci.6b00062