Kriegelstein, M.; Profous, D.; Přibylka, A.; Lyčka, A.; Cankař, P.
Limitations of Trifluoromethylbenzoimidazolylbenzoic Acid as a Chiral Derivatizing Agent to Assign Absolute Configuration for β-Chiral Aminoalcohols
ACS Omega 2022, 7 (15), 12734–12746. DOI: 10.1021/acsomega.1c07234
Supiková, K.; Kosinová, A.; Vavruša, M.; Kopliková, L.; Francois, A.; Pospíšil, J.; Zatloukal, M.; Wever, R.; Hartog, A.; Grúz, J.
Sulfated phenolic acids in plants
Planta 2022, 255 (na), 124 (1-12). DOI: 10.1007/s00425-022-03902-6
Cankařová, N.; Nemec, I.; Krchňák, V.
p-TSA-Mediated Four-Component Reaction: One-Step Access to Mesoionic 1H-Imidazol-3-ium-4-olates, Direct NHC Precursors
Adv. Synth. Catal. 2022, 364 (-), 2996-3003. DOI: 10.1002/adsc.202200398
Dak, M.; Šlachtová, V.; Šebela, M.; Bazgier, V.; Berka, K.; Smiejkowska, N.; Oorts, L.; Cappoen, D.; Brulíková, L.*
Novel heterocyclic hydroxamates as inhibitors of the mycobacterial zinc metalloprotease Zmp1 to probe its mechanism of function
Eur. J. Med. Chem. 2022, 244 (-), 114831 (1-15). DOI: 10.1016/j.ejmech.2022.114831
Toman, D.; Cankař, P.
Synthesis of Unsymmetrical 1,1’-Bibenzimidazoles via an N-Amination Reaction Forming the Key N-N Bond
ChemistrySelect 2022, 7 (38), e202203144. DOI: doi.org/10.1002/slct.202203144
Králová, P.; Žáková, K.; Pospíšilová, L.; Soural, M.
Synthesis of 2,3-Disubstituted Quinoline-4-carbonitriles through Truce–Smiles Rearrangement of Phenacyl-4-nitrobenzenesulfonamides
Eur. J. Org. Chem. 2022, 2022 (28), 31-34. DOI: https://doi.org/10.1002/ejoc.202200531
Borková, L.; Frydrych, I.; Vránová, B.; Jakubcová, N.; Lišková, B.; Gurská, S.; Džubák, P.; Pavliš, P.; Hajdúch, M.; Urban, M.
Lupane derivatives containing various aryl substituents in the position 3 have selective cytostatic effect in leukemic cancer cells including resistant phenotypes
Eur. J. Med. Chem. 2022, 244 (N/A), 114850. DOI: 10.1016/j.ejmech.2022.114850
Hodoň, J.; Frydrych, I.; Trhlíková, Z.; Pokorný, J.; Borková, L.; Benická, S.; Vlk, M.; Lišková, B.; Kubíčková, A.; Medvedíková, M.; Pisár, M.; Sarek, J.; Das, V.; Ligasová, A.; Koberna, K.; Džubák, P.; Hajdúch, M.; Urban, M.
Triterpenoid pyrazines and pyridines – synthesis, cytotoxicity, mechanism of action, preparation of prodrugs
Eur. J. Med. Chem. 2022, 243 (N/A), 114777. DOI: 10.1016/j.ejmech.2022.114777
Tomanová, M.; Kozlanská, K.; Jorda, R.; Jedinák, L.; Havlíková, T.; Řezníčková, E.; Peřina, M.; Klener, P.; Dolníková, A.; Cankař, P.; Kryštof, V.
Synthesis and Structural Optimization of 2,7,9-Trisubstituted purin-8-ones as FLT3-ITD Inhibitors
Int. J. Mol. Sci. 2022, 23 (24), 16169. DOI: 10.3390/ijms232416169
Porubský, M.; Řezníčková, E.; Křupková, S.; Kryštof, V.; Hlaváč, J.
Development of fluorescent dual-FRET probe for simultaneous detection of caspase-8 and caspase-9 activities and their relative quantification
Bioorg. Chem. 2022, 129 (-), 106151. DOI: 10.1016/j.bioorg.2022.106151