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Triple-FRET multi-purpose fluorescent probe for three-protease detection
RSC Advances 2022, 12 (44), 28780-28787. DOI: 10.1039/d2ra05125g
Zhang, H.X.; Daněk, O.; Makarov, D.; Rádl, S.; Kim, D.; Ledvinka, J.; Vychodilová, K.; Hlaváč, J.; Lefebre, J.; Denis, M.; Rademacher, C.; Ménová, P.
Drug-like Inhibitors of DC-SIGN Based on a Quinolone Scaffold
ACS Med. Chem. Letters 2022, 13 (6), 935-942. DOI: 10.1021/acsmedchemlett.2c00067
Okorochenkov, S.; Škrott, Z.; Majera, D.; Porubský, M.; Mistrik, M.; Hlaváč, J.
BODIPY-aza-indole derivate complex as a selective fluorescent sensor for autolysosomes detection
Sens. Actuator B-Chem. 2022, 351 (-), 130941. DOI: 10.1016/j.snb.2021.130941
Hernychová, L.; Alexandri, E.; Tzakos, A. G.; Zatloukalová, M.; Primikyri, A.; Gerothanassis, I. P.; Uhrik, L.; Šebela, M.; Kopečný, D.; Jedinák, L.; Vacek, J.
Serum albumin as a primary non-covalent binding protein for nitro-oleic acid
Int. J. Biol. Macromol. 2022, 2022 (203) (4), 116-129. DOI: 10.1016/j.ijbiomac.2022.01.050
Sobczak, K.; Rudnicki, K.; Jedinak, L.; Zatloukalova, M.; Vacek, J.; Poltorak, L.
Oleic and nitro-oleic acid behavior at an electrified water-1,2-dichloroethane interface
J. Mol. Liquids 2022, 2022 (365) (N/A), 120110(1-6). DOI: 10.1016/j.molliq.2022.120110
Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094 (1-10). DOI: 10.1016/j.ejmech.2020.113094
Ručilová, V.; Świerczek, A.; Vanda, D.; Funk, P. ; Lemrová, B.; Gawalska, A.; Bucki, A.; Nowak, B.; Zadrożna, M.; Pociecha, K.; Soural, M.; Wyska, E.; Pawłowski, M.; Chłoń-Rzepa, G.; Zajdel, P.
New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases
Eur. J. Med. Chem. 2021, 209 (-), 112854(1-18). DOI: 10.1016/j.ejmech.2020.112854
Chasák, J.; Šlachtová, V.; Urban, M.; Brulíková, L.*
Squaric acid analogues in medicinal chemistry
Eur. J. Med. Chem. 2021, 209 (-), 112872 (1-23). DOI: 10.1016/j.ejmech.2020.112872
Kriegelsteinová, P.; Lemrová, B.; Ručilová, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021, 363 (4), 1112-1119. DOI: 10.1002/adsc.202001403
Vanda, D.; Canale, V.; Chaumont-Dubel, S.; Kurczab, R.; Satała, G.; Koczurkiewicz, P.; Krawczyk, M.; Pietruś, W.; Blicharz, K.; Pękala, E.; Bojarski, A.; Popik, P.; Marin, P.; Soural, M.; Zajdel, P.
Imidazopyridine-based 5-HT6 receptor neutral antagonists: impact of N1-benzyl and N1-phenylsulfonyl fragments on different receptor conformational state
J. Med. Chem. 2021, 64 (2), 1180-1196. DOI: 10.1021/acs.jmedchem.0c02009