Tkadlecová, M.; Lemrová, B.; Soural, M.
Synthesis of Polysubstituted Pyridines and Pyrazines via Truce-Smiles Rearrangement of Amino Acid-based 4-Nitrobenzenesulfonamides
J. Org. Chem. 2023, 88 (5), 3228-3237. DOI: 10.1021/acs.joc.2c03025
Ondrová, K.; Zůvalová, I.; Vyhlídalová, B.; Krasulová, K.; Miková, E.; Vrzal, R.; Nádvorník, P.; Nepal, B.; Kortagere, S.; Kopečná, M.; Kopečný, D.; Šebela, M.; Rastinejad, F.; Pu, H.; Soural, M.; Rolfes, K. M.; Haarmann-Stemmann, T.; Li, H.; Mani, S.; Dvořák, Z.
Monoterpenoid aryl hydrocarbon receptor allosteric antagonists protect against ultraviolet skin damage in female mice
Nat. Commun. 2023, 14 (-), 2728-2743. DOI: 10.1038/s41467-023-38478-6
Sládeková, L.; Zgarbová, E.; Vrzal, R.; Vanda, D.; Soural, M.; Jakubcová, K.; Vázquez-Gómez, G.; Vondráček, J.; Dvořák, Z.
Switching on/off aryl hydrocarbon receptor and pregnane X receptor activities by chemically modified tryptamines
Toxicol. Lett. 2023, 387 (-), 63-75. DOI: doi.org/10.1016/j.toxlet.2023.09.012
Králová, P.; Soural, M.
Synthesis of Polycyclic Tetrahydroisoquinolines and Tetrahydrobenzo[d]azepines from Polymer-Supported Allylglycine
J. Org. Chem. 2022, 87 (8), 5242–5256. DOI: 10.1021/acs.joc.2c00039
Lemrová, B.; Maloň, M.; Soural, M.
Efficient Synthesis of Pentasubstituted Pyrroles via intramolecular C-arylation
Org. Biomol. Chem. 2022, 20 (-), 3811-3816. DOI: 10.1039/D2OB00536K
Řezníčková, E.; Krajčovičová, S.; Peřina, M.; Kovalová, M.; Soural, M.; Kryštof, V.
Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC)
Eur. J. Med. Chem. 2022, 243 (-), 114792. DOI: 10.1016/j.ejmech.2022.114792
Králová, P.; Žáková, K.; Pospíšilová, L.; Soural, M.
Synthesis of 2,3-Disubstituted Quinoline-4-carbonitriles through Truce–Smiles Rearrangement of Phenacyl-4-nitrobenzenesulfonamides
Eur. J. Org. Chem. 2022, 2022 (28), 31-34. DOI: https://doi.org/10.1002/ejoc.202200531
Ručilová, V.; Świerczek, A.; Vanda, D.; Funk, P. ; Lemrová, B.; Gawalska, A.; Bucki, A.; Nowak, B.; Zadrożna, M.; Pociecha, K.; Soural, M.; Wyska, E.; Pawłowski, M.; Chłoń-Rzepa, G.; Zajdel, P.
New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases
Eur. J. Med. Chem. 2021, 209 (-), 112854(1-18). DOI: 10.1016/j.ejmech.2020.112854
Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094 (1-10). DOI: 10.1016/j.ejmech.2020.113094
Kriegelsteinová, P.; Lemrová, B.; Ručilová, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021, 363 (4), 1112-1119. DOI: 10.1002/adsc.202001403