Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094 (1-10). DOI: 10.1016/j.ejmech.2020.113094
Kriegelsteinová, P.; Lemrová, B.; Ručilová, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021, 363 (4), 1112-1119. DOI: 10.1002/adsc.202001403
Vanda, D.; Canale, V.; Chaumont-Dubel, S.; Kurczab, R.; Satała, G.; Koczurkiewicz, P.; Krawczyk, M.; Pietruś, W.; Blicharz, K.; Pękala, E.; Bojarski, A.; Popik, P.; Marin, P.; Soural, M.; Zajdel, P.
Imidazopyridine-based 5-HT6 receptor neutral antagonists: impact of N1-benzyl and N1-phenylsulfonyl fragments on different receptor conformational state
J. Med. Chem. 2021, 64 (2), 1180-1196. DOI: 10.1021/acs.jmedchem.0c02009
Maková, B.; Mik, V.; Lišková, B.; González, G.; Vítek, D.; Medvedíková, M.; Monfort, B.; Ručilová, V.; Kadlecová, A.; Khirsariya, P.; Barreiro, Z. G.; Havlíček, L.; Zatloukal, M.; Soural, M.; Paruch, K.; D’Autréaux, B.; Hajdúch, M.; Strnad, M.; Voller J.
Cytoprotective activities of kinetin purine isosteres
Bioorg. Med. Chem. 2021, 33 (-), 115993. DOI: 10.1016/j.bmc.2021.115993
Králová, P.; Soural, M.
Reagent-Based Diversity-Oriented Synthesis of Triazolo[1,5-a][1,4]diazepine Derivatives from Polymer-Supported Homoazidoalanine
J. Org. Chem. 2021, 86 (12), 7963-7974. DOI: 10.1021/acs.joc.1c00293
Krajčovičová, S.; Danišková, A.; Bendová, K.; Nový, Z.; Soural, M.; Petřík, M.
[68Ga]Ga-DFO-c(RGDyK): synthesis and evaluation of its potential for tumor imaging in mice
Int. J. Mol. Sci. 2021, 22 (14), 7391(1-16). DOI: 10.3390/ijms22147391
Králová, P.; Maloň, M.; Pospíšil, J.; Soural, M.
Rearrangement of Threonine and Serine-Based N-(3-Phenylprop-2-yn-1-yl) Sulfonamides Yields Chiral Pyrrolidin-3-ones
J. Org. Chem. 2020, 85 (2), 985-993. DOI: 10.1021/acs.joc.9b02932
Horák, R.; Kořistek, K.; Šamšulová, V. .; Slaninová, L.; Grepl, M.; Kvapil, L.; Funk, P.; Hradil P.; Soural, M.
Structural analogues of quinoline alkaloids: Straightforward route to [1,3]dioxolo[4,5-c]quinolines with antibacterial properties
J. Heterocyclic Chem. 2020, 57 (4), 1605-1615. DOI: 10.1002/jhet.3886
Jorda, R.; Krajčovičová, S.; Králová, P.; Soural, M.; Kryštof, V.
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome
Eur. J. Med. Chem. 2020, 204 (-), 112636. DOI: 10.1016/j.ejmech.2020.112636
Filová, E.; Tonar, Z.; Lukášová, V.; Buzgo, M.; Litvinec, A.; Rampichová, M.; Beznoska, J.; Plencner, M.; Staffa, A.; Daňková, J.; Soural, M.; Chvojka, J.; Malečková, A.; Králíčková, M.; Amler, E.
Hydrogel containing anti-CD44-labeled microparticles, guide bone tissue formation in osteochondral defects in rabbits
Nanomaterials 2020, 10 (8), 1504-1521. DOI: 10.3390/nano10081504