Vyhledat publikace
Chasák, J.; Berka, K.; Bazgier, V.; Cappoen, D.; Brulíková, L.
Squaric acid derivatives as new potential antituberculosis agents
56th Advances in Organic, Bioorganic and Pharmaceutical Chemistry, November 10 – 12, 2022, Špindlerův mlýn, poster .
Dak, M.; Šlachtová, V.; Šebela, M.; Bazgier, V.; Berka, K.; Smiejkowska, N.; Oorts, L.; Cappoen, D.; Brulíková, L.
Novel heterocyclic hydroxamates as inhibitors of the mycobacterial zinc metalloprotease Zmp1
56th Advances in Organic, Bioorganic and Pharmaceutical Chemistry, November 10 – 12, 2022, Špindlerův mlýn, poster .
Cankařová, N.; Nemec, I.; Krchňák, V.
Unprecedented Four-Component Reaction: One-Step Access to Mesoionic 1H-Imidazol-3-ium-5-olates, Direct NHC Precursors
56th Advances in Organic, Bioorganic and Pharmaceutical Chemistry, November 10 – 12, 2022, Špindlerův Mlýn, poster .
Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094 (1-10). DOI: 10.1016/j.ejmech.2020.113094
Ručilová, V.; Świerczek, A.; Vanda, D.; Funk, P. ; Lemrová, B.; Gawalska, A.; Bucki, A.; Nowak, B.; Zadrożna, M.; Pociecha, K.; Soural, M.; Wyska, E.; Pawłowski, M.; Chłoń-Rzepa, G.; Zajdel, P.
New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases
Eur. J. Med. Chem. 2021, 209 (-), 112854(1-18). DOI: 10.1016/j.ejmech.2020.112854
Chasák, J.; Šlachtová, V.; Urban, M.; Brulíková, L.*
Squaric acid analogues in medicinal chemistry
Eur. J. Med. Chem. 2021, 209 (-), 112872 (1-23). DOI: 10.1016/j.ejmech.2020.112872
Kriegelsteinová, P.; Lemrová, B.; Ručilová, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021, 363 (4), 1112-1119. DOI: 10.1002/adsc.202001403
Vanda, D.; Canale, V.; Chaumont-Dubel, S.; Kurczab, R.; Satała, G.; Koczurkiewicz, P.; Krawczyk, M.; Pietruś, W.; Blicharz, K.; Pękala, E.; Bojarski, A.; Popik, P.; Marin, P.; Soural, M.; Zajdel, P.
Imidazopyridine-based 5-HT6 receptor neutral antagonists: impact of N1-benzyl and N1-phenylsulfonyl fragments on different receptor conformational state
J. Med. Chem. 2021, 64 (2), 1180-1196. DOI: 10.1021/acs.jmedchem.0c02009
Urban, M.; Šlachtová, V.; Brulíková, L.*
Small organic molecules targeting the energy metabolism of Mycobacterium tuberculosis
Eur. J. Med. Chem. 2021, 212 (-), 113139 (1-17). DOI: 10.1016/j.ejmech.2020.113139
Maková, B.; Mik, V.; Lišková, B.; González, G.; Vítek, D.; Medvedíková, M.; Monfort, B.; Ručilová, V.; Kadlecová, A.; Khirsariya, P.; Barreiro, Z. G.; Havlíček, L.; Zatloukal, M.; Soural, M.; Paruch, K.; D’Autréaux, B.; Hajdúch, M.; Strnad, M.; Voller J.
Cytoprotective activities of kinetin purine isosteres
Bioorg. Med. Chem. 2021, 33 (-), 115993. DOI: 10.1016/j.bmc.2021.115993