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Krajcovicova, S.; Spring, D. R.
Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late-Stage Functionalisation
Angew. Chem. Int. Ed. 2023, 62 (-), e202307782. DOI: 10.1002/anie.202307782

Tomanová, M.; Vaňková, I.; Toman, D.; Přibylka, A.; Nemec, I.; Cankař, P.
Axially Chiral Sulfonic Acids for Brønsted Acid Catalysis: 8-Benzoimidazolylnaphthalene-1-sulfonic Acids and Their Derivatives
J. Org. Chem. 2023, 88 (13), 9265–9276. DOI: 10.1021/acs.joc.3c00818

King, T.; Walsh, S.; Kapun, M.; Wharton, T.; Krajcovicova, S.; Glossop, M.; Spring, D.
Disulfide re-bridging reagents for single-payload antibody-drug conjugates
Chem. Commun. 2023, 59 (-), 9868-9871. DOI: 10.1039/D3CC02980H

Šlachtová, V.; Casaretto, N.; Brulíková, L.; Six, Y.*
Bicyclic N-dihalocyclopropylamide derivatives as precursors of nitrogen-containing fused polycyclic systems
Org. Biomol. Chem. 2023, 21 (31), 6325-6341. DOI: 10.1039/D3OB00643C

Šamšulová, V.; Šedivá, M.; Kóňa, J. ; Klaudiny, J.; Poláková, M.
A Comparison of the Antibacterial Efficacy of Carbohydrate Lipid‐like (Thio)Ether, Sulfone, and Ester Derivatives against Paenibacillus larvae
Molecules 2023, 28 (-), 2516. DOI: doi.org/10.3390/molecules28062516

Sládeková, L.; Zgarbová, E.; Vrzal, R.; Vanda, D.; Soural, M.; Jakubcová, K.; Vázquez-Gómez, G.; Vondráček, J.; Dvořák, Z.
Switching on/off aryl hydrocarbon receptor and pregnane X receptor activities by chemically modified tryptamines
Toxicol. Lett. 2023, 387 (-), 63-75. DOI: doi.org/10.1016/j.toxlet.2023.09.012

Chasák, J.; Oorts, L.; Dak, M.; Šlachtová, V.; Bazgier, V.; Berka, K.; De Vooght, L.; Smiejkowska, N.; Van Calster, K.; Van Moll, L.; Cappoen, D.; Cos, P.; Brulíková, L.*
Expanding the squaramide library as mycobacterial ATP synthase inhibitors: innovative synthetic pathway and biological evaluation
Bioorg. Med. Chem. 2023, 95 (-), 117504(1-18). DOI: 10.1016/j.bmc.2023.117504

Jessica Iegre, ‡ Sona Krajcovicova, ‡ Anders Gunnarsson, Lisa Wissler, Helena Käck, Anna Luchniak, Stefan Tångefjord, Frank Narjes and David R. Spring
A cell-active cyclic peptide targeting the Nrf2/Keap1 protein–protein interaction
Chem. Sci. 2023, 14 (-), 10800-10805. DOI: 10.1039/D3SC04083F

Králová, P.; Soural, M.
Synthesis of Polycyclic Tetrahydroisoquinolines and Tetrahydrobenzo[d]azepines from Polymer-Supported Allylglycine
J. Org. Chem. 2022, 87 (8), 5242–5256. DOI: 10.1021/acs.joc.2c00039

Řezníčková, E.; Krajčovičová, S.; Peřina, M.; Kovalová, M.; Soural, M.; Kryštof, V.
Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC)
Eur. J. Med. Chem. 2022, 243 (-), 114792. DOI: 10.1016/j.ejmech.2022.114792