Vyhledat publikace
Kolařík, M.; Santarém, N.; Cordeiro-da-Silva, A.; Tavares, J.; Novák, M.; Rydlová, V.; Korábečný, J.; Brulíková, L.*
Exploring the Structural Requirements of Fluorinated Benzylidene-Thiazolidinediones for Selective Antitrypanosomal Activity
Eur. J. Med. Chem. 2027, 321 (-), 119382 (1-21). DOI: 10.1016/j.ejmech.2026.119382
Liška, A.; Chrenko, D.; Zatloukalová, M.; Klíma, J.; Papoušková, B.; Kabeláč, M.; Ludvík, J.; Pospíšil, J.; Vacek, J.
Redox Behaviour of Nitro-Fatty Acids and Their Ester
Electrochimica Acta 2026, 545 (n/a), 147698 (p. 1-12). DOI: 10.1016/j.electacta.2025.147698
Kralova, P.; Rehulka, J.; Grychowska, K.; Ivanova, A.; Liskova, B.; Krajcovicova, S.; Gurska, S.; Hajduch, M.; Lemrova, B.; Zakova, K.; Rucilova, V.; Hruba, K.; Mjartanova, T.; Palova, T.; Sedlackova, K.; Katrusakova, H.; Mokshyna, O.; Lamaty, F.; Leoniec, D.; Uweh, E.; Walczak, M.; Polishchuk, P.; Zajdel, P.; Dzubak, P.; Soural, M.
Design, Synthesis and Biological Evaluation of 1H-Pyrrolo[3,2-c]quinolines as Potent and Selective Anti-tubulin Agents Active against Drug-Resistant Cell Lines
J. Med. Chem. 2026, – (-), accepted. DOI: NA
Biedermann, M. P.; Markos, A.; Warm, I.; Schmitt, A.; Heimgärtner, J.; Lang, K.; Wennemers, H.
The AMI-Isonitrile Ligation 2.0: Fast, Selective, and pH Sensitive
Chem 2026, 12 (2), 102752. DOI: 10.1016/j.chempr.2025.102752
Orság, Š.; Frydrych, I.; Lišková, B.; Gurská, S.; Přibylka, A.; Hodoň, J.; Džubák, P.; Hajdúch, M. Urban, M.
Synthesis and biological evaluation of novel C-30 modified lupane triterpenoids selectively cytotoxic against cancer cells
Eur. J. Med. Chem. 2026, 302 ((-)), 118268. DOI: 10.1016/j.ejmech.2025.118268
Chasák, J.; Vyvlečka, P.; Nemec, I.; Matheeussen, A.; Van Pelt, N.; Cos, P.; Caljon, G.; Kryštof, V.; Brulíková, L.*
Cytotoxicity and Antimicrobial Activity Of GaMF1 Analogues
Chem. Med. Chem. 2026, 21 (4), e202500951 (1-17). DOI: 10.1002/cmdc.202500951
Stehlík, J., Pocklanová, R., Profous, D., Lapčíková, B., Cankař, P., Kvítek, L., Lapčík, Ľ
Innovative Copper-Based Heterogeneous Catalyst for Chan–Lam Cross-Coupling
Catalysts 2026, 16 (I), 94(1-14). DOI: https://doi.org/10.3390/catal16010094
Profous, D.; Cankařová, N.; Enengl, J.; Soji, S.; Rinner, U.; Jurečka, P.; Cankař, P.
Second-Generation Synthesis and Analytical Application of TBBA for Chiral Analysis of Amino Acids and Oligopeptides by 1H and 19F NMR Spectroscopy
J. Org. Chem. 2026, 91 (5), 2065-2073. DOI: 10.1021/acs.joc.5c02693
Valenta, M.; Stýskala, J.
Chemical Modification of 2,6,9-Trisubstituted Purine CDK Inhibitors: tert-Butylation at N7/N9 and Access to 2,6,7-Trisubstituted Analogs
ACS Omega 2026, 11 (16), 23833-23844. DOI: 10.1021/acsomega.5c10284
Bachořík, J.; Frydrych, I.; Gurská, S.; Dostál, Š.; Pokorný, J.; Džubák, P.; Hajdúch, M.; Urban, M.
New Synthetic Approach to C‑30 Ethers, Esters, and Amines of Betulin Using the Mitsunobu Reaction and Biological Evaluation of the Products
ACS Omega 2026, 11 (16), 24564-24579. DOI: 10.1021/acsomega.6c00716