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Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094. DOI: 10.1016/j.ejmech.2020.113094

Ručilová, V.; Świerczek, A.; Vanda, D.; Funk, P. ; Lemrová, B.; Gawalska, A.; Bucki, A.; Nowak, B.; Zadrożna, M.; Pociecha, K.; Soural, M.; Wyska, E.; Pawłowski, M.; Chłoń-Rzepa, G.; Zajdel, P.
New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases
Eur. J. Med. Chem. 2021, 209 (-), 112854. DOI: 10.1016/j.ejmech.2020.112854

Chasák, J.; Šlachtová, V.; Urban, M.; Brulíková, L.
Squaric acid analogues in medicinal chemistry
Eur. J. Med. Chem. 2021, 209 (-), 112872 (1-23). DOI: 10.1016/j.ejmech.2020.112872

Kriegelsteinová, P.; Lemrová, B.; Ručilová, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021, 363 (4), 1112-1119. DOI: 10.1002/adsc.202001403

Vanda, D.; Canale, V.; Chaumont-Dubel, S.; Kurczab, R.; Satała, G.; Koczurkiewicz, P.; Krawczyk, M.; Pietruś, W.; Blicharz, K.; Pękala, E.; Bojarski, A.; Popik, P.; Marin, P.; Soural, M.; Zajdel, P.
Imidazopyridine-based 5-HT6 receptor neutral antagonists: impact of N1-benzyl and N1-phenylsulfonyl fragments on different receptor conformational state
J. Med. Chem. 2021, 64 (2), 1180-1196. DOI: 10.1021/acs.jmedchem.0c02009

Urban, M.; Šlachtová, V.; Brulíková, L.
Small organic molecules targeting the energy metabolism of Mycobacterium tuberculosis
Eur. J. Med. Chem. 2021, 212 (-), 13139 (1-17). DOI: 10.1016/j.ejmech.2020.113139

Maková, B.; Mik, V.; Lišková, B.; González, G.; Vítek, D.; Medvedíková, M.; Monfort, B.; Ručilová, V.; Kadlecová, A.; Khirsariya, P.; Barreiro, Z. G.; Havlíček, L.; Zatloukal, M.; Soural, M.; Paruch, K.; D’Autréaux, B.; Hajdúch, M.; Strnad, M.; Voller J.
Cytoprotective activities of kinetin purine isosteres
Bioorg. Med. Chem. 2021, 33 (-), 115993. DOI: 10.1016/j.bmc.2021.115993

Iakovenko, R.; Hlaváč, J.
Visible light-mediated metal-free double bond deuteration of substituted phenylalkenes
Green. Chem. 2021, in presss (-), -. DOI: 10.1039/D0GC03081C

Gonzalez, G.; Hodoň, J.; Kazakova, A.; D’Acunto, C. W.; Kaňovský, P.; Urban, M.; Strnad, M.
Novel pentacyclic triterpenes exhibiting strong neuroprotective activity in SH-SY5Y cells in salsolinol- and glutamate-induced neurodegeneration models
Eur. J. Med. Chem. 2021, 213 (n/a), 113168. DOI: 10.1016/j.ejmech.2021.113168

Chasák, J.; Brulíková, L.
Polymer-supported synthesis of various pteridinones and pyrimidodiazepinones
Molecules 2021, 26 (6), 1603 (1-21). DOI: 10.3390/molecules26061603