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Tkadlecová, M.; Lemrová, B.; Soural, M.
Synthesis of Polysubstituted Pyridines and Pyrazines via Truce-Smiles Rearrangement of Amino Acid-based 4-Nitrobenzenesulfonamides
J. Org. Chem. 2023, 88 (5), 3228-3237. DOI: 10.1021/acs.joc.2c03025

Cankařová, N.; Krchňák, V.
Regioselective Cyclic Iminium Formation of Ugi Advanced Intermediates: Rapid Access to 3,4-Dihydropyrazin-2(1H)-ones and Other Diverse Nitrogen-Containing Heterocycles
Molecules 2023, 28 (7), 3062 (1-17). DOI: 10.3390/molecules28073062

Ondrová, K.; Zůvalová, I.; Vyhlídalová, B.; Krasulová, K.; Miková, E.; Vrzal, R.; Nádvorník, P.; Nepal, B.; Kortagere, S.; Kopečná, M.; Kopečný, D.; Šebela, M.; Rastinejad, F.; Pu, H.; Soural, M.; Rolfes, K. M.; Haarmann-Stemmann, T.; Li, H.; Mani, S.; Dvořák, Z.
Monoterpenoid aryl hydrocarbon receptor allosteric antagonists protect against ultraviolet skin damage in female mice
Nat. Commun. 2023, 14 (-), 2728-2743. DOI: 10.1038/s41467-023-38478-6

Zebrowski, P.; Rösel, K.; Chrenko, D.; Pospíšil, J.; Waser, M.
Enantioselective beta-selective addition of isoxazolidin-5-ones to allenoates catalyzed by quaternary ammonium salts
Synthesis 2023, 55 (11), 1706-1713. DOI: 10.1055/a-1948-5493

Krajcovicova, S.; Spring, D. R.
Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late-Stage Functionalisation
Angew. Chem. Int. Ed. 2023, e202307782 (-), -. DOI: 10.1002/anie.202307782

Tomanová, M.; Vaňková, I.; Toman, D.; Přibylka, A.; Nemec, I.; Cankař, P.
Axially Chiral Sulfonic Acids for Brønsted Acid Catalysis: 8-Benzoimidazolylnaphthalene-1-sulfonic Acids and Their Derivatives
J. Org. Chem. 2023, 88 (13), 9265–9276. DOI: 10.1021/acs.joc.3c00818

King, T.; Walsh, S.; Kapun, M.; Wharton, T.; Krajcovicova, S.; Glossop, M.; Spring, D.
Disulfide re-bridging reagents for single-payload antibody-drug conjugates
Chemical Communications 2023, (-), -. DOI: 10.1039/D3CC02980H

Šlachtová, V.; Casaretto, N.; Brulíková, L.; Six, Y.*
Bicyclic N-dihalocyclopropylamide derivatives as precursors of nitrogen-containing fused polycyclic systems
Org. Biomol. Chem. 2023, 21 (31), 6233-6428. DOI: 10.1039/D3OB00643C

Šamšulová, V.; Šedivá, M.; Kóňa, J. ; Klaudiny, J.; Poláková, M.
A Comparison of the Antibacterial Efficacy of Carbohydrate Lipid‐like (Thio)Ether, Sulfone, and Ester Derivatives against Paenibacillus larvae
Molecules 2023, 28 (-), 2516. DOI: doi.org/10.3390/molecules28062516

Sládeková, L.; Zgarbová, E.; Vrzal, R.; Vanda, D.; Soural, M.; Jakubcová, K.; Vázquez-Gómez, G.; Vondráček, J.; Dvořák, Z.
Switching on/off aryl hydrocarbon receptor and pregnane X receptor activities by chemically modified tryptamines
Toxicol. Lett. 2023, 387 (-), 63-75. DOI: doi.org/10.1016/j.toxlet.2023.09.012