Vyhledat publikace
Porubsky,M . Hlaváč, J.
The fluorescent derivative of 5,5-difluoro-7,9-dimethyl-5H-4,4,5,4-dipyrrolo[1,2-c:2′,1′-f][1,3,2]diazaborinin-3-amine
užitný vzor , 32033 , Katedra organické chemie, 2018.
Burglova, K.; Petráček, M.; Přichystalová, H.; Hradil, P.; Soural, M.; Hlaváč, J.
3-Hydroxy-2-phenylquinoline-4(1H)-one derivatives with increased solubility, the method of their preparation and use
patent , 307534 , Ústav molekulární a translační medicíny, 2018.
Volná, T.;Motyka, K.; Hlaváč. J.
RP-HPLC determination of dissociation constant using solely aqueous mobile phase
J. Pharm. Biomed. Anal. 2017, 134 (-), 143-148. DOI: 10.1016/j.jpba.2016.11.038
La-Venia, A.; Ventosa, P. A.; Krchňák, V.
Peptidomimetics via Iminium Chemistry on Solid Phase: Single, Fused, and Bridged Heterocycles
Top. Heterocycl. Chem. 2017, 49 (-), 105-126. DOI: 10.1007/7081_2015_194
Krajčovičová, S.; Gucký, T.; Hendrychová, D.; Kryštof, V.; Soural, M.
A Stepwise Approach for the Synthesis of Folic Acid Conjugates with Protein Kinases Inhibitors
J. Org. Chem. 2017, 82 (24), 13530-13541. DOI: 10.1021/acs.joc.7b02650
Ručil, T.; Trávníček, Z.; Cankař, P.
Ring-Opening Reactions of the N-4-Nosyl Hough–Richardson Aziridine with Nitrogen Nucleophiles
J. Org. Chem. 2017, 82 (1), 723-730. DOI: 10.1021/acs.joc.6b01942
Jedinák, L.; Zátopková, R.; Zemánková, H.; Šustková, A.; Cankař, P.
The Suzuki–Miyaura Cross-Coupling Reaction of Halogenated Aminopyrazoles: Method Development, Scope, and Mechanism of Dehalogenation Side Reaction
J. Org. Chem. 2017, 82 (1), 157-169. DOI: 10.1021/acs.joc.6b02306
Králová, P.; Fülöpová, V.; Maloň, M.; Volná, T.; Popa, I.; Soural, M.
Stereoselective polymer-supported synthesis of morpholine and thiomorpholine-3-carboxylic acid derivatives
ACS Comb. Sci. 2017, 19 (3), 173-180. DOI: 10.1021/acscombsci.6b00178
Burglova, K.; Okorochenkov, S.; Budesinsky, M.; Hlavac, J.
Efficient Method for Aromatic-Aldehyde Oxidation by Cleavage of Their Hydrazones Catalysed by Trimethylsilanolate
Eur. J. Org. Chem. 2017, 2017 (2), 389–396. DOI: 10.1002/ejoc.201601238
Šidová, V.; Zoufalý, P.; Pokorný, J.; Džubák, P.; Hajdúch, M.; Popa, I.; Urban, M
Cytotoxic conjugates of betulinic acid and substituted triazoles prepared by Huisgen Cycloaddition from 30-azidoderivatives
PLoS ONE 2017, 12 (2), e0171621. DOI: 10.1371/journal.pone.0171621