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Autorské časopisecké publikace

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Bon, D. J.-Y. D.; Mander, L. N.; Lan, P.
Syntheses of Gibberellins A15 and A24, the Key Metabolites in Gibberellin Biosynthesis
J. Org. Chem. 2018, 83 (12), 6566-6572. DOI: 10.1021/acs.joc.8b00876

Burglova, K.; Hlavac, J.
Application of Trimethylsilanolate Alkali Salts in Organic Synthesis
Synthesis 2018, 50 (6), 1199-1208. DOI: 10.1055/s-0037-1609202

Burglova, K.; Rylova, G.; Markos, A.; Prichystalova, H.; Soural, M.; Petracek, M.; Medvedikova, M.; Tejral, G.; Sopko, B.; Hradil, P.; Dzubak, P.; Hajduch, M.; Hlavac, J.
Identification of Eukaryotic Translation Elongation Factor 1-​α 1 Gamendazole-​Binding Site for Binding of 3-​Hydroxy-​4(1H)​-​quinolinones as Novel Ligands with Anticancer Activity
J. Med. Chem. 2018, 61 (7), 3027-3036. DOI: 10.1021/acs.jmedchem.8b00078

Králová, P.; Soural, M.
Synthesis of 2-Alkylsulfonyl-imidazoles with Three Diversity Positions from Immobilized alpha-Acylamino Ketones
ACS Comb. Sci. 2018, 20 (8), 467-471. DOI: 10.1021/acscombsci.8b00075

Kralová, P.; Ručilová, V.; Soural, M.
Polymer-Supported Syntheses of Heterocycles Bearing Oxazine and Thiazine Scaffolds
ACS Comb. Sci. 2018, 20 (9), 529–543. DOI: 10.1021/acscombsci.8b00076

Lasák, P.; Motyka, K.; Kryštof, V.; Stýskala, J.
Synthesis, Bacteriostatic and Anticancer Activity of Novel Phenanthridines Structurally Similar to Benzo[c]phenanthridine Alkaloids
Molecules 2018, 23 (9), 2155/1-2155/24. DOI: 10.3390/molecules23092155

Schütznerová, E.; Přibylka, A.; Krchňák, V.
Nα-Amino acid containing privileged structures: design, synthesis and use in solid-phase peptide synthesis
Org. Biomol. Chem. 2018, 16 (29), 5359-5362. DOI: 10.1039/c8ob01485j

Schütznerová, E.; Oliver, A. G.; Přibylka, A.; Krchňák, V.
Solid‐Phase Synthesis of Tetramic Acid via Resin‐Bound Enol Ethers as a Privileged Scaffold in Drug Discovery
Adv. Synt.Catal. 2018, 360 (19), 3693-3699. DOI: 10.1002/adsc.201800645

Gimenez-Navarro, V.; Krchňák, V.
Traceless Solid-Phase Synthesis of [6,7,8 + 5,6,7]-Fused Molecular Frameworks
Molecules 2018, 23 (5), 1090/1-1090/12. DOI: 10.3390/molecules23051090

Přibylka, A.; Krchňák, V.
An alkyne rod to constrain a peptide backbone in an extended conformation
Eur. J. Org. Chem. 2018, 2018 (34), 4709-4715. DOI: 10.1002/ejoc.201800979