Sydenham J. D. ; Seki, H.; Krajcovicova, S.; Schober, T.; Zeng, L.; Deingruber, T. ; Spring D. R.
Site-Selective Peptide Functionalisation Mediated via Vinyl-Triazine Linchpins
Chem. Commun. 2024, 60 (-), 706-709. DOI: 10.1039/D3CC05213C
Krajcovicova, S.
Ideas Behind the Tryptophan-Mediated Petasis Reaction (TMPR) Concept for Peptide Stapling
ChemMedChem 2024, 19 (-), e202400148. DOI: https://doi.org/10.1002/cmdc.202400148
Krajcovicova, S.*; Spring, D. R.
Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late-Stage Functionalisation
Angew. Chem. Int. Ed. 2023, 62 (-), e202307782. DOI: 10.1002/anie.202307782
King, T.; Walsh, S.; Kapun, M.; Wharton, T.; Krajcovicova, S.; Glossop, M.; Spring, D. R.
Disulfide re-bridging reagents for single-payload antibody-drug conjugates
Chem. Commun. 2023, 59 (-), 9868-9871. DOI: 10.1039/D3CC02980H
Iegre, J.‡; Krajcovicova, S.‡; Gunnarsson, A.; Wissler, L.; Kaeck, H.; Luchniak, A.; Tangefjord, S.; Narjes, F.; Spring, D. R.
A cell-active cyclic peptide targeting the Nrf2/Keap1 protein–protein interaction
Chem. Sci. 2023, 14 (-), 10800-10805. DOI: 10.1039/D3SC04083F
Řezníčková, E.; Krajčovičová, S.; Peřina, M.; Kovalová, M.; Soural, M.; Kryštof, V.
Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC)
Eur. J. Med. Chem. 2022, 243 (-), 114792. DOI: 10.1016/j.ejmech.2022.114792
Krajčovičová, S.; Jorda, R.; Vanda, D..; Soural, M.; Kryštof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem. 2021, 211 (-), 113094 (1-10). DOI: 10.1016/j.ejmech.2020.113094
Krajčovičová, S.; Hlaváč, J.; Vychodilová, K.
Polymer-supported synthesis of N-substituted anthranilates as the building blocks for preparation of N-arylated 3-hydroxyquinolin-4(1H)-ones
RSC Advances 2021, 24 (-), 9362-9365. DOI: 10.1039/D1RA01308D
Krajčovičová, S.; Danišková, A.; Bendová, K.; Nový, Z.; Soural, M.; Petřík, M.
[68Ga]Ga-DFO-c(RGDyK): synthesis and evaluation of its potential for tumor imaging in mice
Int. J. Mol. Sci. 2021, 22 (14), 7391(1-16). DOI: 10.3390/ijms22147391
Jorda, R.; Krajčovičová, S.; Králová, P.; Soural, M.; Kryštof, V.
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome
Eur. J. Med. Chem. 2020, 204 (-), 112636. DOI: 10.1016/j.ejmech.2020.112636